发明名称 NOVEL COMPOUND, PROCESS FOR PRODUCING THE SAME, AND ANTITUMOR AGENT.
摘要 <p>A pyridonecarboxylic acid derivative represented by general formula (a) or a salt thereof, a process for producing the compounds, and an antitumor agent containing the same as the active ingredient, wherein R1 represents hydrogen, halogen, etc.; R2 represents carboxy, etc.; R3 represents hydrogen, etc.; A represents nitrogen or CH; m represents 1 or 2; Y represents an eliminable group or a group represented by general formula (b); R4 represents hydrogen or lower alkyl; Z represents hydrogen, lower alkyl, etc.; R5 represents hydrogen, lower alkyl, etc.; n represents 0 or 1; and p represents 1, 2, 3 or 4.</p>
申请公布号 MX9606331(A) 申请公布日期 1997.03.29
申请号 MX19960006331 申请日期 1995.06.06
申请人 DAINIPPON PHARMACEUTICAL CO. LTD. 发明人 KYOJI TOMITA;KATSUMI CHIBA;SHIGEKI KASHIMOTO;KOH-ICHIRO SHIBAMORI;YASUNORI TSUZUKI
分类号 A61K31/435;A61K31/4747;A61K31/505;A61P35/00;C07D417/04;C07D417/14;C07D471/04;(IPC1-7):C07D417/04 主分类号 A61K31/435
代理机构 代理人
主权项
地址