发明名称 |
NOVEL PYRIDONECARBOXYLIC ACID DERIVATIVES OR THEIR SALTS, AND ANTIBACTERIAL AGENTS CONTAINING THE SAME AS THEIR EFFECTIVE COMPONENTS |
摘要 |
Pyridonecarboxylic acid derivatives represented by general formula (1) or their salts, wherein R1 represents hydrogen or a carboxyl protecting group; R2 represents hydroxy, lower alkoxy or optionally substituted amino; R3 represents hydrogen or halogeno; R4 represents hydrogen or halogeno; R5 represents optionally halogenated or substituted saturated cyclic amino; R6 represents hydrogen, halogeno, nitro or optionally protected amino; X, Y and Z may be the same or different and each represents nitrogen, -CH= or -CR7= wherein R7 represents lower alkyl, halogeno or cyano, provided that at least one of X, Y and Z represents nitrogen; and W represents nitrogen or -CR8= wherein R8 represents hydrogen, halogeno or lower alkyl.
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申请公布号 |
CA2232728(A1) |
申请公布日期 |
1997.03.27 |
申请号 |
CA19962232728 |
申请日期 |
1996.09.20 |
申请人 |
WAKUNAGA PHARMACEUTICAL CO., LTD. |
发明人 |
AMANO, HIROTAKA;KURAMOTO, YASUHIRO;HAYASHI, NORIHIRO;YAZAKI, AKIRA;NIINO, YOSHIKO;OHSHITA, YOSHIHIRO;HIRAO, YUZO |
分类号 |
C07D213/74;A61K31/00;A61K31/435;A61K31/4375;A61K31/44;A61K31/4427;A61K31/444;A61K31/47;A61K31/4709;A61K31/495;A61K31/496;A61K31/505;A61K31/506;A61P31/00;A61P31/04;C07D205/04;C07D213/61;C07D213/72;C07D213/73;C07D213/75;C07D213/80;C07D213/85;C07D215/06;C07D239/30;C07D239/42;C07D239/46;C07D239/48;C07D401/04;C07D401/12;C07D401/14;C07D471/04;C07K5/062;(IPC1-7):C07D401/04;C07D519/00;A61K38/05;A61K38/06;C07K5/083;C07D413/14;C07D417/14;A61K31/535;A61K31/54;A61K31/55 |
主分类号 |
C07D213/74 |
代理机构 |
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代理人 |
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