发明名称 NOVEL PYRIDONECARBOXYLIC ACID DERIVATIVES OR THEIR SALTS, AND ANTIBACTERIAL AGENTS CONTAINING THE SAME AS THEIR EFFECTIVE COMPONENTS
摘要 Pyridonecarboxylic acid derivatives represented by general formula (1) or their salts, wherein R1 represents hydrogen or a carboxyl protecting group; R2 represents hydroxy, lower alkoxy or optionally substituted amino; R3 represents hydrogen or halogeno; R4 represents hydrogen or halogeno; R5 represents optionally halogenated or substituted saturated cyclic amino; R6 represents hydrogen, halogeno, nitro or optionally protected amino; X, Y and Z may be the same or different and each represents nitrogen, -CH= or -CR7= wherein R7 represents lower alkyl, halogeno or cyano, provided that at least one of X, Y and Z represents nitrogen; and W represents nitrogen or -CR8= wherein R8 represents hydrogen, halogeno or lower alkyl.
申请公布号 CA2232728(A1) 申请公布日期 1997.03.27
申请号 CA19962232728 申请日期 1996.09.20
申请人 WAKUNAGA PHARMACEUTICAL CO., LTD. 发明人 AMANO, HIROTAKA;KURAMOTO, YASUHIRO;HAYASHI, NORIHIRO;YAZAKI, AKIRA;NIINO, YOSHIKO;OHSHITA, YOSHIHIRO;HIRAO, YUZO
分类号 C07D213/74;A61K31/00;A61K31/435;A61K31/4375;A61K31/44;A61K31/4427;A61K31/444;A61K31/47;A61K31/4709;A61K31/495;A61K31/496;A61K31/505;A61K31/506;A61P31/00;A61P31/04;C07D205/04;C07D213/61;C07D213/72;C07D213/73;C07D213/75;C07D213/80;C07D213/85;C07D215/06;C07D239/30;C07D239/42;C07D239/46;C07D239/48;C07D401/04;C07D401/12;C07D401/14;C07D471/04;C07K5/062;(IPC1-7):C07D401/04;C07D519/00;A61K38/05;A61K38/06;C07K5/083;C07D413/14;C07D417/14;A61K31/535;A61K31/54;A61K31/55 主分类号 C07D213/74
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