ACYLATED AMINOALKANEIMIDAZOLES AND TRIAZOLES, PROCESS FOR PREPARING THEREOF, AND PHARMACOLOGICAL COMPOSITION CONTAINING SAID COMPOUNDS

摘要

FIELD: medicine. SUBSTANCE: claimed invention describes azole compounds of formula (I):wherein said substituents have different meanings which are in free form or in salt form. Said compounds are prepared by acylation or opening of aziridine and oxazole ring. Said compounds are useful as pharmaceutical agents, especially as selective inhibitors of hydroxylases of 25-hydroxyvitamin D3 in treating diseases associated with proliferation and differentiation of tissues dependent on vitamin D. EFFECT: improved properties of the pharmaceutical composition.