N-HETEROCYCLIC COMPOUNDS, INTERMEDIATE PRODUCTS USED TO PREPARE THEM, AGENTS CONTAINING THEM AND THEIR USE IN ANTIFUNGAL APPLICATIONS

摘要

Disclosed are N-heterocyclic compounds of the general formula (I) as well as their salts and N-oxides, in which the variables are as follows, and the R<1> to R<26> groups, independently of one another, are hydrogen, cyano, nitro, halogen, aminocarbonyl, methylsulfonyl, alkyl, alkyl halide, alkoxy, alkoxy halide, alkylthio, alkoxyalkyl, alkoxycarbonyl, or optionally substituted aryl, aryloxy or heteroaryl; m is 0, 1 or 2; Alk is optionally substituted 1,2-ethylidene or 1,3-propylidene; X is oxygen, sulfur or -N(R<5>)-, R<5> being hydrogen, alkyl or cycloalkyl; Q is optionally substituted aryl, heteroaryl, cycloalkyl, cycloalkenyl or arylalkyl; excepting (a) compounds V1 to V26 in which A = A1 and R<4> = H, (b) compound I in which A is the N-oxide of A1, with R<1>, R<2>, R<3>, R<4> = H, m = 2, Alk = 1,2-ethylidene, X = -O-, Q = phenyl, and (c) compounds I in which A = A2 and at the same time m = 0. Disclosed also are intermediate products used to prepare these compounds, agents containing them and their use in antifungal applications.