发明名称 Substituted N-heteroaryl-1,2-diaminocyclobutene-3,4-dione compounds
摘要 The compounds of formula I are smooth muscle relaxants: <IMAGE> (I) wherein R1 is hydrogen, alkyl, cycloalkyl, alkanoyl, alkylsulfonyl, aroyl, arylalkenoyl, arylsulfonyl, arylalkanoyl or arylalkylsulfonyl; R2 is hydrogen, alkyl or cyclic or bicyclic alkyl; A is selected from the following: <IMAGE> <IMAGE> <IMAGE> <IMAGE> <IMAGE> <IMAGE>
申请公布号 US5605909(A) 申请公布日期 1997.02.25
申请号 US19960601632 申请日期 1996.02.14
申请人 AMERICAN HOME PRODUCTS CORPORATION 发明人 BUTERA, JOHN A.;ANTANE, SCHUYLER A.;HIRTH, BRADFORD H.
分类号 C07D239/42;A61K31/135;A61K31/275;A61K31/415;A61K31/4184;A61K31/44;A61K31/4406;A61K31/4409;A61K31/47;A61K31/472;A61P13/02;A61P15/00;A61P43/00;C07C225/20;C07C255/58;C07C255/60;C07D213/38;C07D213/75;C07D215/38;C07D217/02;C07D231/56;C07D235/04;(IPC1-7):C07D213/02 主分类号 C07D239/42
代理机构 代理人
主权项
地址