| 摘要 |
This patent describes the derivative of 2-iminobenzothiazoline with a general formula (I), where R1 represents a polyfluoralkoxy or polyfluoralkyl group and R2 represents the group called -CH2-(CH(R4)n-R3, where R3 represents a dialkylamino group, piperidine group, 1-pyrolidine group, merkaptol group, acylthio group, alkyltio group, alkylsulphynil group or alkylsulphonyl group and the symbol called R4 represents a hydrogen atom or an alkyl group and n is a number 0 or 1, or R2 represents a group with a general formula (A), where the symbol R1 is of the above mentioned meaning. This patent also contains a description of enantiomers closed to this derivative with an asymmetric centre and the salts of this derivative created with the use of organic or inorganic acids, while alkyl groups and alkyl and alkaoxyl residues closed to the other groups contain carbon atoms (1 up to 4) having a direct or a branched chain and the acyl groups contain 2 up to 4 carbon atoms. The description of procedures related to the preparation of the above mentioned derivative, together with the pharmaceutical preparation containing this derivative, is a part of this patent too.
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