发明名称 HETEROARYL DIOL ACIDS AS LEUKOTRIENE ANTAGONISTS
摘要 Compounds of formula (I) are antagonists of the actions of leukotrienes. These compounds are useful as anti-asthmatic, anti-allergic, anti-inflammatory, and cytoprotective agents. They are also useful in treating angina, cerebral spasm, glomerular nephritis, hepatitis, endotoxemia, uveitis, and allograft rejection.
申请公布号 WO9640638(A1) 申请公布日期 1996.12.19
申请号 WO1996US08446 申请日期 1996.06.03
申请人 MERCK FROSST CANADA INC.;GAREAU, YVES;LABELLE, MARC;DUFRESNE, CLAUDE;YERGEY, JAMES;CHAURET, NATHALIE;NICOLI-GRIFFITH, DEBORAH;TRIMBLE, LAIRD;XU, XIN 发明人 GAREAU, YVES;LABELLE, MARC;DUFRESNE, CLAUDE;YERGEY, JAMES;CHAURET, NATHALIE;NICOLI-GRIFFITH, DEBORAH;TRIMBLE, LAIRD;XU, XIN
分类号 C07D215/14;A61K31/44;A61K31/47;A61P1/16;A61P7/00;A61P9/08;A61P9/10;A61P11/08;A61P13/02;A61P15/00;A61P29/00;A61P37/06;A61P37/08;A61P43/00;C07D215/18;C07D495/04;(IPC1-7):C07D215/18;A61K31/435 主分类号 C07D215/14
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