发明名称 Cyclic peptide antifungal agents
摘要 <p>Provided are pharmaceutical formulations, and methods of inhibiting fungal and parasitic activity using a compound of formula I &lt;CHEM&gt; where: R', R", R"', R&lt;x1&gt;, R&lt;x2&gt;, R&lt;y1&gt;, R&lt;y2&gt;, R&lt;y3&gt; R&lt;y4&gt;, and R&lt;0&gt; are as defined hereinabove; and R&lt;2&gt; is &lt;CHEM&gt; or &lt;CHEM&gt; R&lt;3&gt; is &lt;CHEM&gt; or &lt;CHEM&gt; R&lt;3a&gt; is C1-C6 alkyl or C1-C6 alkoxy; R&lt;3b&gt; and R&lt;3c&gt; are independently phenyl or naphthyl; R&lt;3d&gt; is C1-C12 alkyl, C1-C12 alkoxy or -O-(CH2)m-ÄO-(CH2)nÜp-O-(C1-C12 alkyl); m is 2, 3 or 4; n is 2, 3 or 4; p is 0 or 1; or a pharmaceutically acceptable salt thereof.i</p>
申请公布号 EP0744406(A2) 申请公布日期 1996.11.27
申请号 EP19960303603 申请日期 1996.05.21
申请人 ELI LILLY AND COMPANY 发明人 LAGRANDEUR, LISA MARIE HAMMOND;RODRIGUEZ, MICHAEL JOHN;ZWEIFEL, MARK JAMES
分类号 A61K38/00;A61P31/04;A61P31/10;A61P33/00;C07K1/113;C07K7/56;(IPC1-7):C07K7/56;A61K38/12 主分类号 A61K38/00
代理机构 代理人
主权项
地址