发明名称 |
NOVEL SERINE PROTEASE INHIBITORS: DERIVATIVES OF ISOTHIAZOLIDIN-3-ONE-1,1 DIOXIDE AND 3-OXO-1,2,5-THIADIAZOLIDINE-1,1-DIOXIDE |
摘要 |
Isothiazolidin-3-one-1,1 dioxide, 3-oxo-1,2,5-thiadiazolidine-1,1,-dioxide and derivatives thereof, reduce or inhibit the activity of serine proteases. Such compounds are useful as anti-inflammatory and anti-metastatic agents. |
申请公布号 |
EP0739338(A1) |
申请公布日期 |
1996.10.30 |
申请号 |
EP19950908003 |
申请日期 |
1995.01.03 |
申请人 |
THE WICHITA STATE UNIVERSITY |
发明人 |
GROUTAS, WILLIAM, C. |
分类号 |
C07D275/02;A61K31/41;A61K31/425;A61K31/433;A61P29/00;A61P35/02;A61P43/00;C07D275/03;C07D275/06;C07D285/10;C07D417/06;C07D521/00;C07F9/6539;(IPC1-7):C07D285/10 |
主分类号 |
C07D275/02 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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