发明名称 ANELLATED beta -CARBOLINES
摘要 Described are compounds of formula (I), wherein A is a 5-6 membered unsaturated ring in which 1-2 C atoms can be substituted by N, O and/or S and which can be substituted with R<5> and R<6>, and the method for preparing them. Because of their affinity for benzodiazepine receptors, the compounds of formula (I) as well as their salts can be used as drugs. They have different intrinsic efficacy (i.e. agonistic, antagonistic and/or inversely agonistic efficacy) with different isoforms of the GABA benzodiazepine receptor.
申请公布号 WO9632392(A1) 申请公布日期 1996.10.17
申请号 WO1996DE00632 申请日期 1996.04.03
申请人 SCHERING AKTIENGESELLSCHAFT;SEIDELMANN, DIETER;HUTH, ANDREAS;OLESEN, PREBEN, H.;OTTOW, ECKHARD;TURNER, JONATHAN;HILLMANN, MARGRIT;COLE, BELINDA 发明人 SEIDELMANN, DIETER;HUTH, ANDREAS;OLESEN, PREBEN, H.;OTTOW, ECKHARD;TURNER, JONATHAN;HILLMANN, MARGRIT;COLE, BELINDA
分类号 A61K31/40;A61K31/435;A61P25/28;C07D471/04;C07D471/14;C07D495/14;C07D498/14;C07D513/14 主分类号 A61K31/40
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