发明名称 |
Synthesis of epibatidine and analogs thereof |
摘要 |
The present invention provides a method to prepare epibatidine or an analog thereof comprising reacting a bicyclic olefin or diene, such as an azanorbornene, with an aryl or heteroaryl halide or triflate in the presence of a catalytic amount of Pd(O) and a formate salt.
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申请公布号 |
US5565573(A) |
申请公布日期 |
1996.10.15 |
申请号 |
US19930150968 |
申请日期 |
1993.11.12 |
申请人 |
IOWA STATE UNIVERSITY RESEARCH FOUNDATION, INC. |
发明人 |
LAROCK, RICHARD C. |
分类号 |
C07D487/08;(IPC1-7):C07D401/04 |
主分类号 |
C07D487/08 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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