SYNTHESIS OF PEPTIDE - AMINOALKYL AMIDES AND PEPTIDE HYDRAZIDES BY THE SOLID PHASE METHOD

摘要

Compounds of the formula I in which A is hydrogen or an amino protective group, B is an amino acid residue, X is alkylene or aralkylene, Y<1>, Y<2>, Y<3> and Y<4> are identical or different and are hydrogen, methyl, methoxy or nitro, V is hydrogen or a carboxyl protective group, W is -[CH2]n- or -O-[CH2]n-, m is 0 or 1, n is 0 to 6 and p is 0 to 5, are prepared as described and used in the solid-phase synthesis.