| 摘要 |
N-heterocyclyl-aryl-sulphonamides of formula (I) and their salts, excluding 4-(methyl, nitro or amino)-N-(2,1,3-benzothiadiazol-5-yl)-benzenesulphonamide are new: -A=B-C=D- is CH=CH-CH=CH in which 1 or 2 CH may be replaced by N; Ar = phenyl or naphthyl, opt. substd. by 1-3 of halo, Q, 2-6C alkenyl, phenyl, phenoxy, NO2, NR4R5, NHCOR4, CF3, OCF3, CN, OR4, COOR4, (CH2)nCOOR4, (CH2)nNR4R5, NCO or NHCONR4R5; R1,R2 and R3 are absent or are H, halo, Q, CF3, NO2, NR4R5, CN, COOR4 or NHCOR4; R4 and R5 = H or Q, or together are CH2(CH2)nCH2; Q = 1-6C alkyl; X = O or S; halo = F, Cl, Br or iodo, n = 1-3. |
