USE OF A PYRUVATE DEHYDROGENASE ACTIVATOR FOR THE TREATMENT OF ISCHAEMIA IN LIMBS
摘要
Agents which inhibit PDH kinase such as dichloroacetic acid, its salts and derivatives are described as being useful in the treatment of ischaemia in limbs. In particular, dichloroacetic acid and its salts are useful in treating intermittent claudification. Pharmaceutical compositions are also described.
申请公布号
WO9628151(A2)
申请公布日期
1996.09.19
申请号
WO1996GB00555
申请日期
1996.03.11
申请人
ZENECA LIMITED;CONSTANTIN-TEODOSIU, DUMITRU;TIMMONS, JAMES, ARCHIBALD;GREENHAFF, PAUL, LEONARD;POUCHER, SIMON, MARTIN
发明人
CONSTANTIN-TEODOSIU, DUMITRU;TIMMONS, JAMES, ARCHIBALD;GREENHAFF, PAUL, LEONARD;POUCHER, SIMON, MARTIN