发明名称 BALANOIDS
摘要 A novel class of therapeutic compounds, denominated Balanoids, is disclosed. Balanoids have protein kinase C inhibitory activity and selectivity among the isoforms of protein kinase C. Balanoids are useful for treatment of diseases related to protein kinase C in animals, especially humans and is especially indicated for treatment of inflammatory diseases.
申请公布号 WO9420062(A3) 申请公布日期 1996.08.15
申请号 WO1994US02283 申请日期 1994.03.02
申请人 NICHOLS, GINA, M. +LF;SPHINX PHARMACEUTICALS CORPORATION;HALL, STEVEN, EDWARD;BALLAS, LAWRENCE, M.;KULANTHAIVEL, PALANIAPPAN;BOROS, CHRISTIE;JIANG, JACK, B.;JAGDMANN, GUNNAR, ERIK, JR.;LAI, YEN-SHI;BIGGERS, CHRISTOPHER, K.;HU, HONG;HALLOCK, YALI;HUGHES, PHILIP, F.;DEFAUW, JEAN, MARIE;LYNCH, MICHAEL, PATRICK;LAMPE, JOHN, WILLIAM, CROSSLEY;MENALDINO, DAVID, STEVEN;HEERDING, JULIA, MARIE;JANZEN, WILLIAM, P.;HOLLINSHEAD, SEAN, PATRICK 发明人 HALL, STEVEN, EDWARD;BALLAS, LAWRENCE, M.;KULANTHAIVEL, PALANIAPPAN;BOROS, CHRISTIE;JIANG, JACK, B.;JAGDMANN, GUNNAR, ERIK, JR.;LAI, YEN-SHI;BIGGERS, CHRISTOPHER, K.;HU, HONG;HALLOCK, YALI;HUGHES, PHILIP, F.;DEFAUW, JEAN, MARIE;LYNCH, MICHAEL, PATRICK;LAMPE, JOHN, WILLIAM, CROSSLEY;MENALDINO, DAVID, STEVEN;HEERDING, JULIA, MARIE;JANZEN, WILLIAM, P.;HOLLINSHEAD, SEAN, PATRICK;NICHOLS, JEFFREY, BAILEY +DI
分类号 C07D333/36;A61K31/165;A61K31/24;A61K31/34;A61K31/341;A61K31/38;A61K31/381;A61K31/415;A61K31/42;A61K31/425;A61K31/44;A61K31/4427;A61K31/443;A61K31/4433;A61K31/445;A61K31/4468;A61K31/495;A61K31/50;A61K31/55;A61P9/00;A61P25/00;A61P29/00;A61P31/12;A61P35/00;A61P43/00;C07C69/734;C07C233/23;C07C233/41;C07C235/48;C07C235/54;C07C235/84;C07C255/52;C07C311/09;C07C325/00;C07D207/14;C07D207/48;C07D211/56;C07D223/12;C07D257/04;C07D307/22;C07D313/04;C07D337/04;C07D401/04;C07D401/12;C07D401/14;C07D403/12;C07D403/14;C07D405/12;C07D405/14;C07D409/12;C07D413/12;C07D413/14;C07D417/12;C07D417/14;C07F9/572 主分类号 C07D333/36
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