| 摘要 |
4-Mercapto-5-sulphonyl-benzoylguanidines of formula (I) and their salts are new. R1 = A, CF3, CH2F, CHF2 or C2F5; R2 = H, A, 3-7C cycloalkyl, Ph or Het; A = 1-6C alkyl; Ph = phenyl (opt. mono-, di- or tri- substd. by A, OA, NH2, NHA, NA2, F, CI, Br and/or CF3); Het = mono- or bi- cyclic, satd., unsatd. or aromatic, N- or C-bonded heterocycle contg. 1-4 N, O and/or S atoms (opt. mono-, di- or tri- substd. by Hal, CF3, A, OH, OA, SH, SA, NH2, NHA, NA2, CN, NO2 and/or carbonyloxy); Hal = F, Cl, Br or I. |
