发明名称 |
3-PYRROLIDINYLTHIO-CARBAPENEM DERIVATIVES AND THEIR ANTIMICROBAL ACTIVITY |
摘要 |
<p>A compound of formula (I), in which R<1> is carboxy, etc., R<2> is hydroxy(lower)alkyl, etc., R<3> is hydrogen or lower alkyl, R<4> is 2(or 3)-methylpyridin-4-ylmethyl, etc., and R<5> is hydrogen or imino-protective group, or pharmaceutically acceptable salts thereof, which is useful as an antimicrobial agent.</p> |
申请公布号 |
EP0722447(A1) |
申请公布日期 |
1996.07.24 |
申请号 |
EP19940927783 |
申请日期 |
1994.09.27 |
申请人 |
FUJISAWA PHARMACEUTICAL CO., LTD. |
发明人 |
MURATA, MASAYOSHI;TSUTSUMI, HIDEO;MATSUDA, KEIJI;HATTORI, KOHJI;NAKAJIMA, TAKASHI |
分类号 |
C07D477/00;A61K31/397;A61K31/40;A61P31/04;C07D477/20;(IPC1-7):C07D477/20;A61K31/41 |
主分类号 |
C07D477/00 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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