The invention provides a process for producing lamotrigine of formula (I) which process comprises subjecting a compound of formula (II), wherein R is CN or CONH2, in an organic solvent, to ultraviolet or visible radiation and, when R is CN, to heat.
申请公布号
WO9620934(A1)
申请公布日期
1996.07.11
申请号
WO1995GB03048
申请日期
1995.12.29
申请人
THE WELLCOME FOUNDATION LIMITED;WINTER, RAYMOND, GEOFFREY;SAWYER, DAVID, ALAN;GERMAIN, ANDREW
发明人
WINTER, RAYMOND, GEOFFREY;SAWYER, DAVID, ALAN;GERMAIN, ANDREW