发明名称 |
PROCESS FOR PRODUCING 2-(2-HYDROXYMETHYLPHENYL)ACETAMIDE DERIVATIVE AND INTERMEDIATE FOR THE PRODUCTION THEREOF |
摘要 |
<p>A process for producing a compound represented by general formula (I) (E-isomer), wherein R<1> and R<2> are the same or different and each represents hydrogen or alkyl; and R represents hydrogen or alkyl which comprises eliminating the protecting group (P) of the hydroxyl group in the compound represented by general formula (II), wherein R<1>, R<2> and R are as defined above; P represents a protecting group of a hydroxyl group; and SIMILAR represents the configuration of an E- or Z-isomer or a mixture thereof; and an intermediate for the production of compound (I).</p> |
申请公布号 |
WO9620164(A1) |
申请公布日期 |
1996.07.04 |
申请号 |
WO1995JP02621 |
申请日期 |
1995.12.21 |
申请人 |
SHIONOGI & CO., LTD.;TAKASE, AKIRA;KAI, HIROYUKI;MURASHI, TAKAMI |
发明人 |
TAKASE, AKIRA;KAI, HIROYUKI;MURASHI, TAKAMI |
分类号 |
C07C69/738;C07C233/56;C07C249/08;C07C249/12;C07C251/48;C07F7/18;(IPC1-7):C07C251/48;C07C43/174;C07D309/12;C07C323/12;C07C235/72;C07C59/90 |
主分类号 |
C07C69/738 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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