发明名称 SUBSTITUTED TETRA- AND PENTAPEPTIDE INHIBITORS OF PROTEIN:FARNESYL TRANSFERASE
摘要 Inhibitors of protein:farnesyl transferase enzyme are described, as well as methods for the preparation and pharmaceutical compositions of the same, which are useful in controlling tissue proliferative diseases, including cancer and restenosis.
申请公布号 WO9617861(A1) 申请公布日期 1996.06.13
申请号 WO1995US14010 申请日期 1995.10.27
申请人 WARNER-LAMBERT COMPANY 发明人 BOLTON, GARY, LOUIS;CAMPBELL, ALFRED;GOWAN, RICHARD;HODGES, JOHN, COOKE;HUPE, DONALD;LEONARD, DANIELE;SAWYER, TOMI;SEBOLT-LEOPOLD, JUDITH;TINNEY, FRANCIS, J.
分类号 A61K38/00;A61P9/00;A61P35/00;C07K5/103;C07K5/117;C07K7/06;C07K14/47;(IPC1-7):C07K5/117;C07K14/82;A61K38/04 主分类号 A61K38/00
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