发明名称 |
Pyrrolidine-containing monomers and oligomers |
摘要 |
Novel pyrrolidine monomers bearing various functional groups are used to prepare oligomeric structures. The pyrrolidine monomers can be joined via standard phosphate linkages including phosphodiester and phosphorothioate linkages. Useful functional groups include nucleobases as well as polar groups, hydrophobic groups, ionic groups, aromatic groups and/or groups that participate in hydrogen-bonding.
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申请公布号 |
US5519134(A) |
申请公布日期 |
1996.05.21 |
申请号 |
US19940180134 |
申请日期 |
1994.01.11 |
申请人 |
ISIS PHARMACEUTICALS, INC. |
发明人 |
ACEVEDO, OSCAR L.;HEBERT, NORMAND |
分类号 |
A61K31/675;A61K31/80;A61P29/00;A61P43/00;C07D207/12;C07D207/32;C07D207/337;C07D207/34;C07D207/46;C07D233/58;C07D233/60;C07D401/06;C07D401/14;C07D403/06;C07D413/06;C07D417/12;C07D473/34;C07D521/00;C07F9/572;C07F9/6509;C07F9/6561;C08G79/02;C08G79/04;(IPC1-7):C07D207/08;C07D207/06;C07D207/10;C07D239/26 |
主分类号 |
A61K31/675 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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