发明名称 MUSCARINE ANTAGONISTS
摘要 Compounds, 1,3-dihydro-1-{1-[piperidin-4-yl]piperidin-4-yl}-2H-benzimidazol-2-ones and 1,3-dihydro-1-{4-amino-1-cyclohexyl}-2H-benzimidazol-2-ones and derivatives thereof, their preparation, method of use and pharmaceutical compositions are described. These compounds are endowed with antimuscarinic activity and are useful in the treatment and/or prevention of myopia (commonly known as nearsightedness).
申请公布号 WO9613262(A1) 申请公布日期 1996.05.09
申请号 WO1995US13710 申请日期 1995.10.24
申请人 MERCK & CO., INC.;THOMPSON, WAYNE, J.;SUGRUE, MICHAEL, F.;RANSOM, RICHARD, W.;MALLORGA, PIERRE, J.;BELL, IAN, M.;SMITH, ANTHONY, M. 发明人 THOMPSON, WAYNE, J.;SUGRUE, MICHAEL, F.;RANSOM, RICHARD, W.;MALLORGA, PIERRE, J.;BELL, IAN, M.;SMITH, ANTHONY, M.
分类号 A61K31/454;A61K31/4545;A61K31/497;A61K31/501;A61K31/506;A61K31/522;A61K31/5377;A61P27/02;A61P43/00;C07D401/04;C07D401/12;C07D401/14;C07D403/12;C07D471/04;(IPC1-7):A61K31/415;A61K31/42;A61K31/425;A61K31/445;A61K31/44;A61K31/505;A61K31/495;A61K31/33;C07D243/04;C07D233/04;C07D263/62;C07D271/00;C07D277/00;C07D275/00;C07D273/02;C07D295/00;C07D211/00;C07D235/04;C07D285/02;C07D239/24 主分类号 A61K31/454
代理机构 代理人
主权项
地址