发明名称 PYRANONE COMPOUNDS USEFUL TO TREAT RETROVIRAL INFECTIONS
摘要 The present invention relates to compounds of formula I and II which are pyran-2-ones, 5,6-dihydro-pyran-2-ones, 4-hydroxy-benzopyran-2-ones, 4-hydroxy-cycloalkyl[b]pyran-2-ones, and derivatives thereof, useful for inhibiting a retrovirus in a mammalian cell infected with said retrovirus.wherein R10 and R20 taken together are:
申请公布号 WO9530670(A3) 申请公布日期 1996.04.25
申请号 WO1995US05219 申请日期 1995.05.04
申请人 THE UPJOHN COMPANY;ROMINES, KAREN, RENE;BUNDY, GORDON, L.;SCHWARTZ, THERESA, M.;TOMMASI, RUBEN, A.;STROHBACH, JOSEPH, WALTER;TURNER, STEVEN, RONALD;THAISRIVONGS, SUVIT;ARISTOFF, PAUL, ADRIAN;JOHNSON, PAUL, D.;SKULNICK, HARVEY, IRVING;SKALETZKI, LOUIS, L.;ANDERSON, DAVID, JOHN;MORRIS, JOEL;GAMMILL, RONALD, B.;LUKE, GEORGE, P. 发明人 ROMINES, KAREN, RENE;BUNDY, GORDON, L.;SCHWARTZ, THERESA, M.;TOMMASI, RUBEN, A.;STROHBACH, JOSEPH, WALTER;TURNER, STEVEN, RONALD;THAISRIVONGS, SUVIT;ARISTOFF, PAUL, ADRIAN;JOHNSON, PAUL, D.;SKULNICK, HARVEY, IRVING;SKALETZKI, LOUIS, L.;ANDERSON, DAVID, JOHN;MORRIS, JOEL;GAMMILL, RONALD, B.;LUKE, GEORGE, P.
分类号 A61K31/365;A61K31/366;A61K31/415;A61K31/425;A61K31/44;A61K31/4427;A61K31/443;A61K31/47;A61K31/4709;A61K31/505;A61K31/506;A61K31/54;A61P31/12;C07D;C07D309/32;C07D309/38;C07D309/40;C07D311/02;C07D311/08;C07D311/74;C07D311/94;C07D401/12;C07D403/12;C07D405/00;C07D405/12;C07D405/14;C07D407/00;C07D409/00;C07D417/00;C07D417/12 主分类号 A61K31/365
代理机构 代理人
主权项
地址