发明名称 |
[1,2,4]TRIAZOLO[4,3-A]QUINOXALINONE DERIVATIVES, THEIR PREPARATION AND USE |
摘要 |
¢1,2,4!triazolo¢4,3-a!quinoxalinone compounds of general formula (I) wherein R1 is POX'X" or alkyl substituted with COX' or POX'X", and X' and X" independently are hydroxy or alkoxy, and R6, R7, R8 and R9 independently are hydrogen; alkyl; halogen; NH2; NO2; CN; CF3 SO2NY'Y" or COZ' wherein Z' is NY'Y" or alkyl and Y' and Y" independently are hydrogen or alkyl; triazolyl; imidazolyl or imidazolyl substituted with phenyl or alkyl, are useful in the treatment of indications caused by hyperactivity of the excitatory neurotransmitters.
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申请公布号 |
CA2200056(A1) |
申请公布日期 |
1996.03.21 |
申请号 |
CA19952200056 |
申请日期 |
1995.09.12 |
申请人 |
NOVO NORDISK A/S |
发明人 |
NIELSEN, FLEMMING ELMELUND |
分类号 |
A61K31/495;A61P1/08;A61P3/08;A61P9/00;A61P25/00;A61P25/08;A61P25/28;A61P29/00;C07D487/04;(IPC1-7):C07F9/547;A61K31/675 |
主分类号 |
A61K31/495 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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