发明名称 Benzoazepinyl compounds as oxytocin and vasopressin antagonists
摘要 PCT No. PCT/JP93/01082 Sec. 371 Date Apr. 20, 1994 Sec. 102(e) Date Apr. 20, 1994 PCT Filed Aug. 3, 1993 PCT Pub. No. WO94/04525 PCT Pub. Date Mar. 3, 1994.Novel benzoheterocyclic compound of the formula (1): <IMAGE> (1) and pharmaceutically acceptable salts thereof, which show excellent anti-vasopressin activity and oxytocin antagonistic activity, and are useful as a vasopressin antagonist or oxytocin antagonist.
申请公布号 US5498609(A) 申请公布日期 1996.03.12
申请号 US19940211887 申请日期 1994.04.20
申请人 OTSUKA PHARMACEUTICAL COMPANY, LIMITED 发明人 OGAWA, HIDENORI;KONDO, KAZUMI;YAMASHITA, HIROSHI;KAN, KEIZO;TOMINAGA, MICHIAKI;YABUUCHI, YOICHI
分类号 C07D401/06;C07D401/14;C07D405/06;C07D409/06;C07D409/14;C07D413/14;C07D417/06;C07D521/00;(IPC1-7):C07D223/16;A61K31/55 主分类号 C07D401/06
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