发明名称 |
Physical form of dihidro-2,3-benzodiazepine derivative |
摘要 |
A physical form of (R)-7-acetyl-5-(4-aminophenyl)-8,9-dihydro-8-methyl-7H-1,3-dioxoloÄ4,5 -hÜÄ2,3Übenzodiazepine of formula I having an X-ray powder diffraction pattern with d spacings at 10.61, 8.83, 6.78, 5.83, 4.13 and 3.74 ANGSTROM . The compound is useful as an AMPA antagonist. <CHEM> R is methyl, X is acetyl and Aryl is p-nitrophenyl.i |
申请公布号 |
EP0699676(A1) |
申请公布日期 |
1996.03.06 |
申请号 |
EP19950306048 |
申请日期 |
1995.08.30 |
申请人 |
ELI LILLY AND COMPANY |
发明人 |
ANDERSON, BENJAMIN ALAN;HANSEN, MARVIN MARTIN;VICENZI, JEFFREY THOMAS;VARIE, DAVID LEE;ZMIJEWSKI, MILTON JOSEPH, JR.;HARKNESS, ALLEN ROBERT |
分类号 |
C07D491/113;A61K31/55;A61P1/08;A61P25/00;A61P25/04;A61P25/06;A61P25/08;A61P25/14;A61P25/16;A61P25/18;A61P25/20;A61P25/22;A61P25/28;A61P27/02;A61P43/00;C07B63/00;C07D243/00;C07D317/00;C07D317/58;C07D491/04;C07D491/056;C07D493/04 |
主分类号 |
C07D491/113 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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