发明名称 Physical form of dihidro-2,3-benzodiazepine derivative
摘要 A physical form of (R)-7-acetyl-5-(4-aminophenyl)-8,9-dihydro-8-methyl-7H-1,3-dioxoloÄ4,5 -hÜÄ2,3Übenzodiazepine of formula I having an X-ray powder diffraction pattern with d spacings at 10.61, 8.83, 6.78, 5.83, 4.13 and 3.74 ANGSTROM . The compound is useful as an AMPA antagonist. <CHEM> R is methyl, X is acetyl and Aryl is p-nitrophenyl.i
申请公布号 EP0699676(A1) 申请公布日期 1996.03.06
申请号 EP19950306048 申请日期 1995.08.30
申请人 ELI LILLY AND COMPANY 发明人 ANDERSON, BENJAMIN ALAN;HANSEN, MARVIN MARTIN;VICENZI, JEFFREY THOMAS;VARIE, DAVID LEE;ZMIJEWSKI, MILTON JOSEPH, JR.;HARKNESS, ALLEN ROBERT
分类号 C07D491/113;A61K31/55;A61P1/08;A61P25/00;A61P25/04;A61P25/06;A61P25/08;A61P25/14;A61P25/16;A61P25/18;A61P25/20;A61P25/22;A61P25/28;A61P27/02;A61P43/00;C07B63/00;C07D243/00;C07D317/00;C07D317/58;C07D491/04;C07D491/056;C07D493/04 主分类号 C07D491/113
代理机构 代理人
主权项
地址