发明名称 |
Neue 6 und 6,8-substituierte 1-[4-(1H-1,2,4-triazol-l-yl-methyl)phenyl] Chinoloncarbonsäuren |
摘要 |
The invention pertains to 6- and 6,8-substituted 1-[4-(1H-1,2,4-triazol-1-yl methyl) phenyl] quinolone carboxylic acids of general formula (I), in which A is hydrogen or methyl, R<1> is phenyl, naphthyl, pyridyl, pyrimidyl or pyrazinyl, optionally substituted up to three times, alike or differently, by nitro, trifluoromethyl, halogen, cyano, hydroxy or by straight-chain or branched alkyl, acyl, alkoxy or alkylthio with up to 8 carbon atoms in each case, and R<2> is hydrogen, fluorine or chlorine. The invention also pertains to methods for preparing them as well as their use as drugs, especially as antiviral agents.
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申请公布号 |
DE4425648(A1) |
申请公布日期 |
1996.01.25 |
申请号 |
DE19944425648 |
申请日期 |
1994.07.20 |
申请人 |
BAYER AG, 51373 LEVERKUSEN, DE |
发明人 |
BENDER, WOLFGANG, DR., 42113 WUPPERTAL, DE;ROEBEN, WOLFGANG, DR., 51467 BERGISCH GLADBACH, DE;PAESENS, ARNOLD, DR., 42781 HAAN, DE;BARTEL, STEPHAN, DR., 51465 BERGISCH GLADBACH, DE |
分类号 |
C07D249/08;C07D521/00;(IPC1-7):C07D401/10;C07D401/14;A61K31/47;C12N7/06 |
主分类号 |
C07D249/08 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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