发明名称 ARYLSULFONAMIDO-SUBSTITUTED HYDROXAMIC ACIDS AS MATRIX METALLOPROTEINASE INHIBITORS
摘要 Compounds of formula (I) wherein R, R1, R2 and Ar are as defined in the specification, have valuable pharmaceutical properties and are effective especially as matrix metalloproteinase inhibitors, for example for the treatment of arthritis. They are prepared in a manner known per se.
申请公布号 WO9600214(A1) 申请公布日期 1996.01.04
申请号 WO1995IB00464 申请日期 1995.06.12
申请人 CIBA-GEIGY AG;MACPHERSON, LAWRENCE, JOSEPH;PARKER, DAVID, THOMAS;JENG, ARCO, YINGCHEU 发明人 MACPHERSON, LAWRENCE, JOSEPH;PARKER, DAVID, THOMAS;JENG, ARCO, YINGCHEU
分类号 A61K31/18;A61K31/00;A61K31/335;A61K31/357;A61K31/38;A61K31/381;A61K31/382;A61K31/40;A61K31/415;A61K31/42;A61K31/425;A61K31/426;A61K31/435;A61K31/44;A61K31/4402;A61K31/4406;A61K31/4409;A61K31/4418;A61K31/4427;A61K31/443;A61K31/445;A61K31/4465;A61K31/4468;A61K31/47;A61K31/535;A61K31/5375;A61K31/5377;A61K31/55;A61P1/00;A61P1/02;A61P1/04;A61P19/10;A61P27/02;A61P29/00;A61P31/12;A61P35/00;A61P37/04;A61P43/00;C07C311/19;C07C311/29;C07C311/42;C07C323/59;C07D207/08;C07D207/09;C07D207/16;C07D211/26;C07D211/28;C07D211/34;C07D211/58;C07D211/66;C07D211/96;C07D213/42;C07D213/71;C07D215/12;C07D223/10;C07D231/12;C07D231/14;C07D233/24;C07D233/64;C07D233/68;C07D233/84;C07D257/04;C07D261/10;C07D277/06;C07D277/20;C07D277/28;C07D277/30;C07D277/36;C07D295/12;C07D295/14;C07D307/16;C07D309/04;C07D309/14;C07D313/18;C07D317/58;C07D317/60;C07D317/62;C07D333/34;C07D333/58;C07D335/02;C07D401/04;C07D401/06;C07D401/12;C07D405/12;C07D413/06;C07D413/12;C07D521/00;(IPC1-7):C07D213/42 主分类号 A61K31/18
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