发明名称 BICYCLING LACTAM INHIBITOR OF INTERLEUKIN-1-BETA CONVERTING ENZYME
摘要 Disclosed are compounds, compositions, and methods for inhibiting interleukin-1 beta protease activity, having formula (A), wherein Y = (a) or (b) or (c), Z = various bicyclic lactams with a bridgehead nitrogen.
申请公布号 WO9533751(A1) 申请公布日期 1995.12.14
申请号 WO1995US07314 申请日期 1995.06.08
申请人 SANOFI WINTHROP, INC. 发明人 DOLLE, ROLAND, E.;CHATURVEDULA, PRASAD, V.;MORGAN ROSS, TINA;SCHMIDT, STANLEY, J.
分类号 C07D487/04;A61K31/535;A61K31/55;A61K38/00;A61P29/00;A61P35/00;A61P37/06;A61P43/00;C07D471/04;C07D513/04;C07K5/02;C07K5/06;C07K5/078;(IPC1-7):C07D487/04;C07D417/04;C07F9/645;C07F9/650;C07F9/553;C07F9/576;A61K31/495;A61K31/435;A61K31/675 主分类号 C07D487/04
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