发明名称 |
Crystalline forms of endo-2,3-dihydro-N-(8-methyl)-8-azabicyclo[3.2.1]oct-3-yl)-2-oxo-1H-benzimidazole-1-carboxamides |
摘要 |
Crystalline and pharmacologically active monohydrates of endo-2,3-dihydro-N-(8-methyl-8-azabicyclo[3.2.1]oct-3-yl)-2-oxo-1H-benzimidazole-1-carboxamide hydrochloride and of endo-3-ethyl-2,3-dihydro-N-(8-methyl-8-azabicyclo[3.2.1]oct-3-yl)-2-oxo-1H-benzimidazole-1-carboxamide hydrochloride.
|
申请公布号 |
US5468758(A) |
申请公布日期 |
1995.11.21 |
申请号 |
US19940264104 |
申请日期 |
1994.06.22 |
申请人 |
BOEHRINGER INGELHEIM ITALIA S.P.A. |
发明人 |
CEREDA, ENZO;EZHAYA, ANTOINE;TURCONI, MARCO;DUBINI, ENRICA;MAFFIONE, GRAZIA |
分类号 |
A61K31/46;A61K31/415;A61K31/4184;A61K31/495;A61P1/00;A61P1/08;A61P25/00;A61P25/04;A61P25/06;A61P25/18;A61P25/22;A61P25/24;A61P25/28;C07D235/32;C07D403/12;C07D451/04;C07D451/12;(IPC1-7):A61K31/46 |
主分类号 |
A61K31/46 |
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|