摘要 |
The present invention relates to compounds of formulae (I) and (II) (see formula I, II) which are pyran-2-ones, 5,6-dihydro-pyran-2-ones, 4-hydroxy-benzopyran-2-one s, 4-hydroxy-cycloalkyl[b]pyran-2-ones, and derivatives thereof, useful for inhibiting a retrovirus in a mammalian cell infected with said retrovirus, wherein R10 an d R20 taken together are formulae (III) and (IV). (see formula III, IV)
|
申请人 |
PHARMACIA & UPJOHN COMPANY |
发明人 |
GAMMILL, RONALD B.;MORRIS, JOEL;JOHNSON, PAUL D.;SKALETZKY, LOUIS L.;ANDERSON, DAVID JOHN;TOMMASI, RUBEN A.;THAISRIVONGS, SUVIT;ARISTOFF, PAUL ADRIAN;ROMINES, KAREN RENE;LUKE, GEORGE P.;SCHWARTZ, THERESA M.;BUNDY, GORDON L.;STROHBACH, JOSEPH WALTER;TURNER, STEVEN RONALD;SKULNICK, HARVEY IRVING |