发明名称 PYRANONE COMPOUNDS USEFUL TO TREAT RETROVIRAL INFECTIONS
摘要 The present invention relates to compounds of formulae (I) and (II) (see formula I, II) which are pyran-2-ones, 5,6-dihydro-pyran-2-ones, 4-hydroxy-benzopyran-2-one s, 4-hydroxy-cycloalkyl[b]pyran-2-ones, and derivatives thereof, useful for inhibiting a retrovirus in a mammalian cell infected with said retrovirus, wherein R10 an d R20 taken together are formulae (III) and (IV). (see formula III, IV)
申请公布号 CA2560489(A1) 申请公布日期 1995.11.16
申请号 CA19952560489 申请日期 1995.05.04
申请人 PHARMACIA & UPJOHN COMPANY 发明人 GAMMILL, RONALD B.;MORRIS, JOEL;JOHNSON, PAUL D.;SKALETZKY, LOUIS L.;ANDERSON, DAVID JOHN;TOMMASI, RUBEN A.;THAISRIVONGS, SUVIT;ARISTOFF, PAUL ADRIAN;ROMINES, KAREN RENE;LUKE, GEORGE P.;SCHWARTZ, THERESA M.;BUNDY, GORDON L.;STROHBACH, JOSEPH WALTER;TURNER, STEVEN RONALD;SKULNICK, HARVEY IRVING
分类号 C07D405/12;A61K31/365;A61K31/366;A61K31/415;A61K31/425;A61K31/44;A61K31/4427;A61K31/443;A61K31/47;A61K31/4709;A61K31/505;A61K31/506;A61K31/54;A61P31/12;C07D;C07D309/32;C07D309/38;C07D309/40;C07D311/02;C07D311/08;C07D311/20;C07D311/74;C07D311/94;C07D401/12;C07D403/12;C07D405/00;C07D405/14;C07D407/00;C07D409/00;C07D417/00;C07D417/12 主分类号 C07D405/12
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