发明名称 |
INTERMEDIATES AND PROCESSES FOR PREPARING BENZOTHIOPHENE COMPOUNDS |
摘要 |
The present invention provides a novel process for preparing a compound of formula I <IMG> I wherein R1 and R2 combine to form C4-C6 polymethylene, -CH2CH(CH3)CH2CH2-, -CH2C(CH3)2CH2CH2-, or -CH2CH2OCH2CH2-; or a pharmaceutically acceptable salt or solvate thereof, comprising a) reacting a compound of formula II <IMG> II with a compound of formula III <IMG> III
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申请公布号 |
CA2145614(A1) |
申请公布日期 |
1995.10.01 |
申请号 |
CA19952145614 |
申请日期 |
1995.03.27 |
申请人 |
ELI LILLY AND COMPANY |
发明人 |
DODGE, JEFFREY A.;STOCKSDALE, MARK G. |
分类号 |
A61K31/38;A61K31/381;A61P3/00;A61P19/10;A61P43/00;C07D333/56;(IPC1-7):C07D409/12;C07D413/12 |
主分类号 |
A61K31/38 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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