发明名称 INTERMEDIATES AND PROCESSES FOR PREPARING BENZOTHIOPHENE COMPOUNDS
摘要 The present invention provides a novel process for preparing a compound of formula I <IMG> I wherein R1 and R2 combine to form C4-C6 polymethylene, -CH2CH(CH3)CH2CH2-, -CH2C(CH3)2CH2CH2-, or -CH2CH2OCH2CH2-; or a pharmaceutically acceptable salt or solvate thereof, comprising a) reacting a compound of formula II <IMG> II with a compound of formula III <IMG> III
申请公布号 CA2145614(A1) 申请公布日期 1995.10.01
申请号 CA19952145614 申请日期 1995.03.27
申请人 ELI LILLY AND COMPANY 发明人 DODGE, JEFFREY A.;STOCKSDALE, MARK G.
分类号 A61K31/38;A61K31/381;A61P3/00;A61P19/10;A61P43/00;C07D333/56;(IPC1-7):C07D409/12;C07D413/12 主分类号 A61K31/38
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