发明名称 |
NAPHTHALENE DERIVATIVES AS PROSTAGLANDIN 12 AGONISTS |
摘要 |
A compound of formula (I) wherein, R1 is carboxy or protected carboxy: R2 is hydrogen, hydroxy or protected hydroxy; R3 is hydrogen, hydroxy, protected hydroxy, etc.; R4 is hydrogen or halogen; A1 is lower alkylene; A2 is bond or lower alkylene; -R5 is (a) (in which R6 is mono(or di or tri)aryl(lower)alkyl and Z is N or CH), etc; and (b) is (c), etc.; and a pharmaceutically acceptable salt thereof which are useful as medicaments.
|
申请公布号 |
CA2185104(A1) |
申请公布日期 |
1995.09.14 |
申请号 |
CA19952185104 |
申请日期 |
1995.03.08 |
申请人 |
FUJISAWA PHARMACEUTICAL CO., LTD |
发明人 |
OKITSU, OSAMU;TANIGUCHI, KIYOSHI;TSUBAKI, KAZUNORI;TABUCHI, SEIICHIRO;HATTORI, KOUJI;NAGANO, MASANOBU |
分类号 |
A61K31/16;A61K31/335;A61K31/336;A61K31/44;A61K31/4418;A61K31/4425;A61K31/50;A61P7/02;A61P9/10;A61P9/12;A61P43/00;C07C69/145;C07C235/40;C07C271/10;C07C271/12;C07C271/24;C07C271/28;C07C271/32;C07C281/02;C07D213/64;C07D237/14;C07D303/12;C07D303/16;(IPC1-7):C07C271/28;C07D405/02;C07F7/10;A61K31/27;C07C271/38;A61K31/695 |
主分类号 |
A61K31/16 |
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|