This invention is directed to hetero-annulated indazoles of formula (I) and namely to 2,5-disubstituted quinolino-, isoquinolino-, phthalazino-, and quinoxalino-annulated indazole-6(2H)-ones and related mono N-oxides. These compounds have been shown to have antitumor activity.
申请公布号
WO9524407(A1)
申请公布日期
1995.09.14
申请号
WO1995US02862
申请日期
1995.03.08
申请人
BOEHRINGER MANNHEIM ITALIA, S.P.A.;KRAPCHO, A., PAUL;MENTA, ERNESTO;OLIVA, AMBROGIO;SPINELLI, SILVANO
发明人
KRAPCHO, A., PAUL;MENTA, ERNESTO;OLIVA, AMBROGIO;SPINELLI, SILVANO