发明名称 AMINO ACID DERIVATIVES AND THEIR USE AS PHOSPHOLIPASE A2 INHIBITORS
摘要 The present invention relates to a novel fatty acid derivative of formula (I) wherein R<1> is acyl group, etc.; R<2> is acyl(lower)alkyl; R<3> is lower alkyl, etc.; R<4> is hydrogen, etc.; and X is -O-, etc.; and a pharmaceutically acceptable salt thereof, which is useful as a medicament; the processes for the preparation of said fatty acid derivative or a salt thereof; a pharmaceutical composition comprising said fatty acid derivative or a pharmaceutically acceptable salt thereof; etc.
申请公布号 WO9519959(A1) 申请公布日期 1995.07.27
申请号 WO1995JP00068 申请日期 1995.01.23
申请人 FUJISAWA PHARMACEUTICAL CO., LTD.;TAKASE, SHIGEHIRO;SHIGEMATSU, NOBUHARU;YOSHIMURA, SEIJI;OKADA, SATOSHI;HEMMI, KEIJI;TANAKA, HIROKAZU;OTSUKA, TAKANAO;TSURUMI, YASUHISA;OKAMOTO, MASANORI;OKUHARA, MASAKUNI;FUKAMI, NAOKI 发明人 TAKASE, SHIGEHIRO;SHIGEMATSU, NOBUHARU;YOSHIMURA, SEIJI;OKADA, SATOSHI;HEMMI, KEIJI;TANAKA, HIROKAZU;OTSUKA, TAKANAO;TSURUMI, YASUHISA;OKAMOTO, MASANORI;OKUHARA, MASAKUNI;FUKAMI, NAOKI
分类号 C07D295/20;A61K31/165;A61K31/18;A61K31/215;A61K31/27;A61K31/415;A61K31/42;A61K31/423;A61K31/425;A61K31/428;A61K31/44;A61K31/4402;A61K31/4406;A61K31/4409;A61K31/4418;A61K31/445;A61K31/47;A61K31/472;A61K31/535;A61K31/5375;A61K31/5377;A61P1/16;A61P3/06;A61P9/00;A61P9/10;A61P11/00;A61P13/02;A61P15/00;A61P17/00;A61P27/02;A61P27/14;A61P27/16;A61P29/00;A61P37/00;A61P37/08;A61P43/00;C07C227/02;C07C227/08;C07C229/22;C07C235/08;C07C235/12;C07C237/04;C07C237/22;C07C271/22;C07C271/54;C07C275/14;C07C275/16;C07C311/19;C07C311/42;C07D207/16;C07D211/60;C07D211/62;C07D213/38;C07D213/40;C07D213/54;C07D213/56;C07D213/75;C07D213/78;C07D213/81;C07D213/82;C07D215/36;C07D215/38;C07D215/44;C07D215/48;C07D217/06;C07D217/26;C07D233/54;C07D233/64;C07D241/14;C07D241/24;C07D241/44;C07D263/58;C07D277/82;C07D295/215;C07D295/22;C07D295/28;C07D317/58;C07D471/04 主分类号 C07D295/20
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