发明名称 METALLOPROTEINASE INHIBITORS
摘要 Matrix metalloproteinase inhibiting compounds of formula (I), wherein X is a CO2H or -CONHOH group; R4 is a phenyl or 5- or 6-membered heteroaryl ring wherein any ring nitrogen atom may be oxidised as an N-oxide, which may be optionally fused to a benzene ring or to a 5-, 6- or 7-membered heterocyclic ring, and wherein any of the rings may be optionally substituted.
申请公布号 CA2181570(A1) 申请公布日期 1995.07.27
申请号 CA19952181570 申请日期 1995.01.20
申请人 BRITISH BIOTECH PHARMACEUTICALS LIMITED 发明人 BECKETT, RAYMOND PAUL;WHITTAKER, MARK;MILLER, ANDREW;MARTIN, FIONNA MITCHELL
分类号 A61K31/16;A61K31/195;A61K31/33;C07C237/22;C07C259/06;C07D213/75;C07D213/89;C07D271/02;C07D277/46;C07D285/04;C07D307/64;C07D333/34;C07D401/12;C07D409/12;(IPC1-7):C07D285/04 主分类号 A61K31/16
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