摘要 |
<p>Tricyclic benzazepine and benzothiazepine derivatives represented by general formula (I) and pharmacologically acceptable salts thereof, wherein Z represents CO, -CR<6>R<7>- or -S(O)n; R represents hydrogen, alkyl, phenylalkyl or a triazole-protective group; and R<1> to R<5> represent each hydrogen, alkyl, alkenyl, alkoxy, amino, oxime or hydroxy. The compounds have an antiallergic activity and hence are useful for treating and preventing allergic diseases.</p> |
申请人 |
MEIJI SEIKA KABUSHIKI KAISHA;OHTSUKA, YASUO;SHISHIKURA, TAKASHI;OGINO, HIROKO;FUSHIHARA, KENICHI;KAWAGUCHI, MAMI;TSUTSUMI, SEIJI;IMAI, MEGUMI;SHITO, KEIKO;TSUCHIYA, KOJI;TANAKA, JUNKO;IWASAKI, TAKAKO;HOSHIKO, SHIGERU;TSURUOKA, TAKASHI |
发明人 |
OHTSUKA, YASUO;SHISHIKURA, TAKASHI;OGINO, HIROKO;FUSHIHARA, KENICHI;KAWAGUCHI, MAMI;TSUTSUMI, SEIJI;IMAI, MEGUMI;SHITO, KEIKO;TSUCHIYA, KOJI;TANAKA, JUNKO;IWASAKI, TAKAKO;HOSHIKO, SHIGERU;TSURUOKA, TAKASHI |