发明名称 TRICYCLIC BENZAZEPINE AND BENZOTHIAZEPINE DERIVATIVES
摘要 <p>Tricyclic benzazepine and benzothiazepine derivatives represented by general formula (I) and pharmacologically acceptable salts thereof, wherein Z represents CO, -CR<6>R<7>- or -S(O)n; R represents hydrogen, alkyl, phenylalkyl or a triazole-protective group; and R<1> to R<5> represent each hydrogen, alkyl, alkenyl, alkoxy, amino, oxime or hydroxy. The compounds have an antiallergic activity and hence are useful for treating and preventing allergic diseases.</p>
申请公布号 WO9518130(A1) 申请公布日期 1995.07.06
申请号 WO1994JP02282 申请日期 1994.12.28
申请人 MEIJI SEIKA KABUSHIKI KAISHA;OHTSUKA, YASUO;SHISHIKURA, TAKASHI;OGINO, HIROKO;FUSHIHARA, KENICHI;KAWAGUCHI, MAMI;TSUTSUMI, SEIJI;IMAI, MEGUMI;SHITO, KEIKO;TSUCHIYA, KOJI;TANAKA, JUNKO;IWASAKI, TAKAKO;HOSHIKO, SHIGERU;TSURUOKA, TAKASHI 发明人 OHTSUKA, YASUO;SHISHIKURA, TAKASHI;OGINO, HIROKO;FUSHIHARA, KENICHI;KAWAGUCHI, MAMI;TSUTSUMI, SEIJI;IMAI, MEGUMI;SHITO, KEIKO;TSUCHIYA, KOJI;TANAKA, JUNKO;IWASAKI, TAKAKO;HOSHIKO, SHIGERU;TSURUOKA, TAKASHI
分类号 C07D249/04;C07D487/04;C07D513/04;(IPC1-7):C07D487/04;A61K31/55 主分类号 C07D249/04
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