发明名称 |
Pyrroloazepine derivatives |
摘要 |
Disclosed herein are pyrroloazepine derivatives having anti- alpha 1 activity and anti-serotonin activity represented by the following formula (I): linear or branched C1-6 alkyl group or a C7-10 aralkyl group, A denotes a linear or branched C2-10 alkylene, alkenylene or alkynylene group, Z stands for O, NOR1 or NOCOR5 in which R1 and R5 is a hydrogen atom or an alkyl, aryl or aralkyl group, and Y means a particular piperidinyl or pyrrolidinyl group; and salts thereof. Their preparation processes are also disclosed.
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申请公布号 |
US5416082(A) |
申请公布日期 |
1995.05.16 |
申请号 |
US19940195019 |
申请日期 |
1994.02.14 |
申请人 |
SUNTORY LIMITED |
发明人 |
MIZUNO, AKIRA;CHO, HIDETSURA;HAMAGUCHI, MIKIKO;TATSUOKA, TOSHIO;ISHIHARA, TAKAFUMI |
分类号 |
A61K31/55;A61P9/00;A61P9/04;A61P9/12;A61P43/00;C07D487/04;(IPC1-7):A61K31/55 |
主分类号 |
A61K31/55 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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