发明名称 16-SUBSTITUTED-4-AZA-ANDROSTANE 5-ALPHA-REDUCTASE ISOZYME 1 INHIBITORS
摘要 Compounds of formula (I) are inhibitors of the 5 alpha -reductase 1 isozyme, and are useful alone, or in combination with a 5 alpha -reductase 2 inhibitor, for the treatment of androgenic sensitive disorders such as acne vulgaris, seborrhea, female hirsutism, male pattern baldness, and benign prostatic hyperplasia.
申请公布号 WO9511254(A1) 申请公布日期 1995.04.27
申请号 WO1994US12071 申请日期 1994.10.21
申请人 MERCK & CO., INC.;DURETTE, PHILIPPE, L.;HAGMANN, WILLIAM, K.;LANZA, THOMAS, J., JR.;SAHOO, SOUMYA, P.;RASMUSSON, GARY, H.;TOLMAN, RICHARD, L.;VON LANGEN, DEREK 发明人 DURETTE, PHILIPPE, L.;HAGMANN, WILLIAM, K.;LANZA, THOMAS, J., JR.;SAHOO, SOUMYA, P.;RASMUSSON, GARY, H.;TOLMAN, RICHARD, L.;VON LANGEN, DEREK
分类号 A61K31/58;A61P5/24;A61P17/14;A61P29/00;C07J73/00;(IPC1-7):C07J73/00 主分类号 A61K31/58
代理机构 代理人
主权项
地址