发明名称 |
Process for production of 2-acetylbenzo[b]thiophene |
摘要 |
A process for production of 2-acetylbenzo[b]thiophene represented by the formula (I): <IMAGE> comprising the steps of: (1) reacting 2-halogenobenzaldehyde represented by the formula (II): <IMAGE> wherein X represents a halogen atom, with a compound represented by the formula (III): HiSjMk wherein M represents an alkali metal, i represents zero or 1, j represents an integer of at least 1, and k represents an integer of 1 or 2, and preferably also with sulfur; and (2) reacting the reaction product with a monohalogenoacetone represented by the formula (IV) <IMAGE> wherein X1 represents a halogen atom.
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申请公布号 |
US5403939(A) |
申请公布日期 |
1995.04.04 |
申请号 |
US19930118184 |
申请日期 |
1993.09.09 |
申请人 |
TAKEDA CHEMICAL INDUSTRIES, LTD. |
发明人 |
YAZAWA, NAOTO;SAITO, YOSHINORI;HIYOSHI, HIDETAKA |
分类号 |
C07D333/56;(IPC1-7):C07D333/56 |
主分类号 |
C07D333/56 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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