发明名称 4-hydroxyphenylthio derivatives, their preparation and their use for the preparation of aminoalkoxyphenylsulphonyl derivatives
摘要 The subject of the invention is 4-hydroxyphenylthio derivatives of general formula: <IMAGE> I in which: R1 and R2, which are identical or different, each represent hydrogen, a methyl or ethyl radical or a halogen atom, R represents a (C1-C6) alkyl, (C3-C6) cycloalkyl or phenyl radical, R3 represents hydrogen or a halogen atom, X represents -O-, -S- or -NR4- in which R4 represents hydrogen or a (C1-C4) alkyl group, useful as synthetic intermediates, especially for the preparation of aminoalkoxyphenylsulphonyl derivatives which are pharmaceutically active compounds.
申请公布号 US5401855(A) 申请公布日期 1995.03.28
申请号 US19930080171 申请日期 1993.06.23
申请人 ELF SANOFI 发明人 GUBIN, JEAN;INION, HENRI
分类号 C07D209/30;C07D307/82;C07D333/62;C07D403/12;C07D405/12;C07D409/12;(IPC1-7):C07D209/30 主分类号 C07D209/30
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