发明名称 POLYAMIDIC ACID DERIVATIVES WITH ANTIGASTRIN ACTIVITY, A METHOD FOR THEIR PREPARATION, AND THEIR PHARMACEUTICAL USE
摘要 New derivatives of glutamic and aspartic acids of formula (I) are described. The compounds are potent receptor antagonists of gastrin at the peripheral level and of cholecystokinin at the level of the central nervous system.
申请公布号 WO9507261(A1) 申请公布日期 1995.03.16
申请号 WO1994EP02983 申请日期 1994.09.07
申请人 ROTTA RESEARCH LABORATORIUM S.P.A.;MAKOVEC, FRANCESCO;PERIS, WALTER;ROVATI, LUCIO, CLAUDIO;ROVATI, LUIGI, ANGELO 发明人 MAKOVEC, FRANCESCO;PERIS, WALTER;ROVATI, LUCIO, CLAUDIO;ROVATI, LUIGI, ANGELO
分类号 C07D215/48;A61K31/40;A61K31/403;A61K31/404;A61K31/435;A61K31/44;A61K31/4427;A61K31/47;A61K38/00;A61P1/04;A61P27/02;C07D209/20;C07D209/54;C07D221/20;C07D401/12;C07D403/12;C07D471/10;C07K5/02;C07K5/078;(IPC1-7):C07D221/20;C07D401/06;C07D209/10;C07K5/08;A61K31/165 主分类号 C07D215/48
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