发明名称 |
PROCESSES AND INTERMEDIATES FOR PHOSPHOROUS-CONTAINING COVALENT LINKAGES |
摘要 |
Synthetic processes are provided wherein substituted silylalkyl phosphoramidites serve as coupling reagents for preparing phosphate, phosphorothionate, and other phosphorus-containing covalent linkages. Also provided are synthetic intermediated useful in such processes.
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申请公布号 |
CA2167671(A1) |
申请公布日期 |
1995.02.09 |
申请号 |
CA19942167671 |
申请日期 |
1994.07.20 |
申请人 |
ISIS PHARMACEUTICALS, INC. |
发明人 |
RAVIKUMAR, VASULINGA;MULVEY, DENNIS;COLE, DOUGLAS L.;COOK, PHILLIP DAN |
分类号 |
C07H19/06;A61K31/70;A61K31/7042;A61K31/7052;A61K31/7064;A61K31/7068;A61K31/7072;A61K31/7076;A61K31/708;A61K31/7088;A61P31/12;A61P35/00;C07F9/146;C07F9/24;C07H19/16;C07H21/00;C07H21/02;C07H21/04;C07H23/00;(IPC1-7):C07H23/00;C07H19/04 |
主分类号 |
C07H19/06 |
代理机构 |
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