发明名称 PHENANTHRENDERIVAT.
摘要 A novel phenanthrene derivative of general formula (1), its salt, a compound further derived therefrom, and its salt; a process for the production thereof; and an interleukin 1 (IL-1) inhibitor containing the derivative as the active ingredient, wherein (a) represents (b) wherein R' represents hydrogen or lower alkyl, (c) wherein R<2> represents hydrogen or lower alkanoyl, or (d) wherein R<2> is as defined above.
申请公布号 DE69106281(D1) 申请公布日期 1995.02.09
申请号 DE1991606281 申请日期 1991.03.05
申请人 OTSUKA PHARMACEUTICAL CO., LTD., TOKIO/TOKYO, JP;OTSUKA PHARMACEUTICAL FACTORY, INC., NARUTO, TOKUSHIMA, JP 发明人 TAKAISHI, YOSHIHISA, TOKUSHIMA-SHI, TOKUSHIMA 770, JP;GOTO, KIYOTO, 57, AZA UMAGOE, AKINOKAMI, SETOCHO, TOKUSHIMA 772, JP;UESAKO, TAKUJI, 51-6, AZA MINAMIKAWAMUKAI, ITANO-GUN, TOKUSHIMA 771-02, JP;KUWAHARA, TOSHIKO, 14-21, NAKANOKOSHI, AZA NAKASE, TOKUSHIMA 771-02, JP;TAKAI, MASAAKI, 62-14, AZA MINAMIKAWAMUKAI, TOKUSHIMA 771-0, JP;ONO, YUKIHISA, 41-18, AZA KAWAKUBO, TAINOHAMA, ITANO-GUN, TOKUSHIMA 771-02, JP;TANIGUCHI, YOSHIHIRO, RA FORE KAWAUCHI 407, TOKUSHIMA-SHI, TOKUSHIMA 770, JP;MANABE, SACHIKO, 463-10, KAGASUNO, KAWAUCHICHO, TOKUSHIMA 770, JP;ASAKUNI, TAKAHIRO, 81, NIBUDOI, OUCHICHO, KANAGAWA 769-26, JP
分类号 C07C49/747;C07C50/34;C07C50/38;C07C62/32;C07C62/34;C07C62/38;C07C69/00;C07C69/007;C07C69/013;C07C69/757;C07D307/77;(IPC1-7):C07C49/747;C07C66/00;C07C69/02;C07C69/95;A61K31/19;A61K31/215 主分类号 C07C49/747
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