发明名称 INHIBITION OF PHOSPHATIDYLINOSITOL 3-KINASE WITH WORTMANNIN AND ANALOGS THEREOF
摘要 of the Invention Wortmannin and certain of its analogs are inhibitors of phosphatidylinositol 3-kinase. The compounds are particularly useful for inhibiting phosphatidylinositol 3-kinase in mammals and for treating phosphatidylinositol 3-kinase-dependent conditions, especially neoplasms, in mammals.
申请公布号 CA2128046(A1) 申请公布日期 1995.01.20
申请号 CA19942128046 申请日期 1994.07.14
申请人 ELI LILLY AND COMPANY;ARIZONA BOARD OF REGENTS (THE) 发明人 BONJOUKLIAN, ROSANNE;POWIS, GARTH;VLAHOS, CHRIS J.
分类号 A61K31/58;A61K31/34;A61K31/343;A61K31/365;A61K31/585;A61P35/00;A61P43/00;C07D307/77;(IPC1-7):A61K31/365 主分类号 A61K31/58
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