| 发明名称 |
Saccharin derivative proteolytic enzyme inhibitors |
| 摘要 |
Compounds having the structural formula <IMAGE> Formula I which inhibit the enzymatic activity of proteolytic enzymes, and processes for preparation thereof, method of use thereof in treatment of degenerative diseases and pharmaceutical compositions thereof are disclosed.
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| 申请公布号 |
US5378720(A) |
申请公布日期 |
1995.01.03 |
| 申请号 |
US19930066805 |
申请日期 |
1993.05.25 |
| 申请人 |
STERLING WINTHROP INC. |
发明人 |
HLASTA, DENNIS J.;ACKERMAN, JAMES H.;MURA, ALBERT J.;DESAI, RANJIT C. |
| 分类号 |
A61K31/425;A61K31/428;A61K31/435;A61K31/445;A61K31/47;A61K31/505;A61K31/519;A61K31/535;A61P1/00;A61P1/18;A61P13/02;A61P15/00;A61P17/00;A61P29/00;A61P43/00;C07D275/06;C07D417/12;C07D471/04;C07D487/04;C07D513/04;(IPC1-7):A61K31/425;C07D417/14 |
主分类号 |
A61K31/425 |
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