发明名称 NOVEL PILOCARPINE DERIVATIVES AND PROCESS FOR THEIR PREPARATION
摘要 The object of the invention are novel bispilocarpates useful in the treatment of glaucoma and having general formula (I), wherein A) Y is hydrogen or the acyl group (II), and W is the group -O-A-O-Z-Y', wherein Y' is hydrogen or the acyl group (III), the groups R and R' having different meanings and may be the same or different and A is an aliphatic or aromatic bridging group, and -Z-Y' is (IV), or B) W is OR, wherein R has the same meaning as above, Y is (V), where R' has the same meaning as above, B means the same as A and Z'-OR' is (VI) or C) W and Y together mean -A-O-Z-C-B-C-, where the symbols have the same meanings as above.
申请公布号 LTIP577(A) 申请公布日期 1994.12.27
申请号 LTIP577 申请日期 1993.05.28
申请人 LEIRAS OY 发明人 JAERVINEN,TOMI;PEURA,PEKKA;SUHONEN,PEKKA;URTTI,ARTO;HANHIJAERVI,HANNU;POHJALA,ESKO
分类号 A61K31/415;A61K31/4164;A61K31/4178;A61P27/02;A61P27/06;C07D233/54;C07D233/58;C07D233/64;C07D405/14 主分类号 A61K31/415
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