发明名称 Indole indazole and benzisoxazole compounds process for preparing them and pharmaceutical compositions containing them
摘要 The invention relates to the compounds of formula (I): <IMAGE> in which: R1 represents a hydrogen or halogen atom, an alkyl, alkoxy, cyano or aminocarbonyl group or any one of the following groups: <IMAGE> -(CH2)m-NH-COR6, -(CH2)m-NH-SO2-R4, <IMAGE> -(CH2)m-NH-CO-NHR4, <IMAGE> -(CH2)m-SO2-NH-R4, -CH=CH-SO2-NH-R4, <IMAGE> in which: m is equal to 1, 2 or 3, n is equal to 0, 1 or 2, T represents a CO or SO2, R4 or R5, which are identical or different, represent a hydrogen atom or an alkyl or phenyl group, R2 represents a hydrogen atom or an alkyl, phenyl or acyl group, R3 represents a hydrogen atom or an alkyl (optionally substituted by a hydroxyl or phenyl group) or alkoxycarbonyl group, -X-Y= represents -N-C=, -N-N= or else <IMAGE> represents -O-N=, to their enantiomers, diastereoisomers and epimers and to their addition salts with a pharmaceutically acceptable acid. Medicaments.
申请公布号 ZA9400709(B) 申请公布日期 1994.09.06
申请号 ZA19940000709 申请日期 1994.02.02
申请人 ADIR ET COMPAGNIE 发明人 GILBERT LAVIELLE;PHILIPPE MAILLOS;OLIVIER MULLER;MICHEL LAUBIE;TONY VERBEUREN;JEAN-JACQUES DESCOMBES
分类号 A61K31/40;A61K31/415;A61P25/04;C07D403/06;C07D403/14;C07D413/06;C07D413/14;C07D419/14 主分类号 A61K31/40
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