发明名称 |
N-(pyrrolo(2,3-d)pyrimidin-3-ylacyl)-glutamic acid derivatives |
摘要 |
N-(Acyl)glutamic acid derivatives in which the acyl group is substituted with 4-hydroxypyrrolo[2,3-d]-pyrimidin-3-yl group are antineoplastic agents. A typical embodiment is N-[4-(2-{4-hydroxy-6-aminopyrrolo-[2,3-d]pyrimidin-3-yl}ethyl)benzoyl]-L-glutamic acid.
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申请公布号 |
US5344932(A) |
申请公布日期 |
1994.09.06 |
申请号 |
US19910674541 |
申请日期 |
1991.03.22 |
申请人 |
TRUSTEES OF PRINCETON UNIVERSITY |
发明人 |
TAYLOR, EDWARD C. |
分类号 |
C07D487/04;(IPC1-7):C07D487/04;A61K31/505 |
主分类号 |
C07D487/04 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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