发明名称 SPIRO-SUBSTITUTED AZACYCLES AS TACHYKININ RECEPTOR ANTAGONISTS
摘要 Disclosed are spiro-substituted azacycles of formula (I), are tachykinin receptor antagonists useful in the treatment of inflammatory diseases, pain or migraine, emesis and asthma. In particular compounds of formula (I) are shown to be neurokinin antagonists.
申请公布号 WO9417045(A1) 申请公布日期 1994.08.04
申请号 WO1994US00819 申请日期 1994.01.25
申请人 MERCK & CO., INC.;HALE, JEFFREY, J.;MACCOSS, MALCOLM;MILLS, SANDER, G.;QI, HONGBO;SHAH, SHRENIK, K. 发明人 HALE, JEFFREY, J.;MACCOSS, MALCOLM;MILLS, SANDER, G.;QI, HONGBO;SHAH, SHRENIK, K.
分类号 A61K31/445;A61P1/08;A61P11/00;A61P25/04;A61P29/00;A61P43/00;C07D221/20;C07D491/10;C07D491/107;C07D495/20;(IPC1-7):C07D221/20 主分类号 A61K31/445
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